Mefloquin® Tablets USP 250mg

Brand Name: Mefloquin® by Taj Pharmaceuticals Ltd.

Premium quality antimalarial medication trusted by healthcare professionals worldwide for the treatment and prevention of malaria.

Key Highlights

  • USP Quality Standards
  • WHO-GMP Certified Manufacturing
  • Export Quality Assurance
  • Stringent Quality Control
  • High Efficacy Rate
  • Long-Lasting Protection
  • Global Regulatory Compliance
  • Competitive Pricing

Composition

Each tablet contains:

  • Mefloquine Hydrochloride USP equivalent to Mefloquine 250mg
  • Excipients: Lactose monohydrate, Croscarmellose sodium, Magnesium stearate

Mechanism of Action

Mefloquin® is a quinoline methanol compound with schizonticidal activity. It acts by forming toxic complexes with free heme that damage membranes and interact with other plasmodial biopolymers. The exact mechanism of action is not fully understood, but it is believed to interfere with heme polymerization, which is essential for parasite survival.

Primary Action

Inhibits heme polymerization in malaria parasites

Secondary Effects

Disrupts parasite membrane function and metabolism

Pharmacology Summary

Parameter Details
Onset of Action 2-4 hours after oral administration
Peak Plasma Concentration 6-23 hours post-dose
Half-life 2-3 weeks
Protein Binding 98.5%
Metabolism Hepatic metabolism

Clinical Benefits

High Cure Rate

Proven efficacy in treating uncomplicated P. falciparum malaria

Long-Lasting

Extended half-life provides prolonged protection

Global Acceptance

WHO-approved and widely used internationally

Quality Assured

Manufactured under strict WHO-GMP guidelines

Why Choose Mefloquin® (Taj Advantage)

🏭 Manufacturing Excellence

State-of-the-art WHO-GMP certified facilities with advanced manufacturing processes

🔬 Quality Assurance

Rigorous quality control at every stage from raw materials to finished product

🌍 Global Standards

Compliance with international pharmacopeial standards and regulatory requirements

📊 Research & Development

Continuous improvement through ongoing research and clinical studies

🤝 Customer Support

Comprehensive medical information and regulatory support services

💰 Competitive Pricing

Cost-effective solution without compromising on quality or efficacy